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2006:234207 BIOSIS
DN
PREV200600228562
TI
peroxisome proliferator-activated receptor-gamma transcriptionally up-regulates hormone-sensitive lipase via the involvement of specificity protein-1.
AU
Deng, Tuo; Shan, Song; Li, Ping-Ping; Shen, Zhu-Fang; Lu, Xian-Ping; Cheng, Jing; Ning, Zhi-Qiang [Reprint Author]
CS
Tsing Hua Univ, Shenzhen Res Inst, Chipscreen Biosci Ltd, Shenzhen 518057, Peoples R China zqning@chipscreen.com
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Endocrinology, (FEB 2006) Vol. 147, No. 2, pp. 875-884. CODEN: ENDOAO. ISSN: 0013-7227.
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Article
LA
English
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Entered STN: 12 Apr 2006 Last Updated on STN: 12 Apr 2006
AB
Both peroxisome proliferator-activated receptor (PPAR)-gamma and hormone-sensitive lipase (HSL) play important roles in lipid metabolism and insulin sensitivity. We demonstrate that expression of the HSL gene is up-regulated by PPAR gamma and PPAR gamma agonists (rosiglitazone and pioglitazone) in the cultured hepatic cells and differentiating preadipocytes. Rosiglitazone treatment also results in up-regulation of the HSL gene in liver and skeleton muscle from an experimental obese rat model, accompanied by the decreased triglyceride content in these tissues. The proximal promoter (-87 bp of the human HSL gene) was found to be essential for PPAR gamma-mediated transactivating activity. This important promoter region contains two GC-boxes and binds the transcription factor specificity protein-1 (Sp1) but not PPAR gamma. The Sp1-promoter binding activity can be endogenously enhanced by PPAR gamma and rosiglitazone, as demonstrated by analysis of EMSA and chromatin immunoprecipitation assay. Mutations in the GC-box sequences reduce the promoter binding activity of Sp1 and the transactivating activity of PPAR gamma. In addition, mithramycin A, the specific inhibitor for Sp1-DNA binding activity, abolishes the PPAR gamma-mediated up-regulation of HSL. These results indicate that PPAR gamma positively regulates the HSL gene expression, and up-regulation of HSL by PPAR gamma requires the involvement of Sp1. Taken together, this study suggests that HSL may be a newly identified PPAR gamma target gene, and up-regulation of HSL may be an important mechanism involved in action of PPAR gamma agonists in type 2 diabetes.
CC
Cytology - Animal 02506 Cytology - Human 02508 Genetics - General 03502 Genetics - Animal 03506 Genetics - Human 03508 Biochemistry studies - Lipids 10066 Enzymes - General and comparative studies: coenzymes 10802 Pathology - Therapy 12512 Metabolism - Metabolic disorders 13020 Nutrition - Malnutrition and obesity 13203 Digestive system - Physiology and biochemistry 14004 Endocrine - General 17002 Endocrine - Pancreas 17008 Muscle - Physiology and biochemistry 17504 Pharmacology - Clinical pharmacology 22005 Pharmacology - Blood and hematopoietic agents 22008 Pharmacology - Cardiovascular system 22010 Pharmacology - Endocrine system 22016 Pediatrics 25000
IT
Major Concepts Molecular Genetics (Biochemistry and Molecular Biophysics); Enzymology (Biochemistry and Molecular Biophysics); Endocrine System (Chemical Coordination and Homeostasis)
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Parts, Structures, & Systems of Organisms liver: digestive system; skeletal muscle: muscular system; preadipocyte; hepatic cell: digestive system
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Diseases type 2 diabetes: endocrine disease/pancreas, metabolic disease Diabetes Mellitus, Non-Insulin-Dependent (MeSH)
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Diseases obesity: nutritional disease Obesity (MeSH)
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Chemicals & Biochemicals triglyceride; peroxisome proliferator-activated receptor-alpha; hormone-sensitive lipase; pioglitazone: antidiabetic-drug; specificity protein 1; mithramycin A: enzyme inhibitor-drug; rosiglitazone: antidiabetic-drug, thrombolytic-drug, hematologic-drug, cardiovascular-drug, vasodilator-drug
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Methods & Equipment immunoprecipitation: laboratory techniques, immunologic techniques; electrophoresis mobility shift assay [EMSA]: electrophoretic techniques, genetic techniques, laboratory techniques
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Miscellaneous Descriptors lipid metabolism; insulin sensitivity
ORGN
Classifier Hominidae 86215 Super Taxa Primates; Mammalia; Vertebrata; Chordata; Animalia Organism Name SMMC-7721 cell line (cell_line): human hepatoma cells CCC-L cell line (cell_line): human fetal liver cells Taxa Notes Animals, Chordates, Humans, Mammals, Primates, Vertebrates
ORGN
Classifier Muridae 86375 Super Taxa Rodentia; Mammalia; Vertebrata; Chordata; Animalia Organism Name Wistar rat (common): newborn Taxa Notes Animals, Chordates, Mammals, Nonhuman Vertebrates, Nonhuman Mammals, Rodents, Vertebrates
RN
9001-62-1 (hormone-sensitive lipase) 111025-46-8 (pioglitazone) 97666-60-9 (mithramycin A) 122320-73-4 (rosiglitazone)
GEN
rat HSL gene [rat hormone-sensitive lipase gene] (Muridae): up-regulation